{"id":2772,"date":"2016-09-15T21:34:12","date_gmt":"2016-09-16T01:34:12","guid":{"rendered":"https:\/\/www.med.unc.edu\/genetics\/perou-and-collaborators-published-in-disease-models-and-mechanisms\/"},"modified":"2018-02-07T11:25:09","modified_gmt":"2018-02-07T16:25:09","slug":"perou-and-collaborators-published-in-disease-models-and-mechanisms","status":"publish","type":"post","link":"https:\/\/www.med.unc.edu\/genetics\/perou-and-collaborators-published-in-disease-models-and-mechanisms\/","title":{"rendered":"Perou and collaborators published in Disease Models and Mechanisms"},"content":{"rendered":"<p><!-- description --><\/p>\n<p class=\"lead\">Charles Perou, PhD, Professor of Genetics and Pathology and Laboratory Medicine and the May Goldman Shaw Distinguished Professor of Molecular Oncology was corresponding author of a study that focused on finding possible drug targets in triple-negative breast cancers.<\/p>\n<div class=\"newsitem\">\n<figure class=\"thumbnail wp-caption alignright\" style=\"width: 260px\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.med.unc.edu\/genetics\/wp-content\/uploads\/sites\/481\/2017\/10\/perou-and-collaborators-published-in-disease-models-and-mechanisms-image2.jpeg\" alt=\"Charles Perou, PhD\" width=\"250\" height=\"333\" \/><figcaption class=\"caption wp-caption-text\">Charles Perou, PhD<\/figcaption><\/figure>\n<\/div>\n<p>The paper, titled \u201cGenomic Profiling of Murine Mammary Tumors Identifies Potential Personalized Drug Targets for p53-Deficient Mammary Cancers\u201d was published in the 01 July 2016 issue of Disease Models and Mechanisms. Along with colleagues from Washington University, University of Albany and Baylor College of Medicine, the Perou laboratory utilized a murine <i>Trp53<\/i>-null mammary transplant tumor model to identify additional drivers and possible drug targets of the triple-negative breast cancer phenotype. Two subsets of transplant tumors resembled human basal-like subtype and DNA-microarray, whole-genome and exome-based sequencing were used to study the secondary genetic aberrations which were compared to human basal-like tumors to identify conserved somatic genetic features. After filtering the candidates (gene deemed essential in at least 5% of human breast cancer cell lines), five potential personalized drug target genes were identified, including <i>Cul4a, Lamp1, Met, Pnpla6 <\/i>and<i> Tubgcp3<\/i>. Inhibition of <i>Met<\/i> using crizotinib caused <i>Met<\/i>-amplified murine tumors to undergo complete regression, identifying <i>Met<\/i> as a promising drug target in the mouse tumor models and highlighting the utility of comparative genomic studies and preclinical models for interrogating tumor signaling pathways.<\/p>\n<p>Link to the article: <a class=\"external-link\" title=\"\" href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/27149990\" target=\"_blank\" rel=\"noopener noreferrer\">http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/27149990<\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Charles Perou, PhD, Professor of Genetics and Pathology and Laboratory Medicine and the May Goldman Shaw Distinguished Professor of Molecular Oncology was corresponding author of a study that focused on finding possible drug targets in triple-negative breast cancers. The paper, titled \u201cGenomic Profiling of Murine Mammary Tumors Identifies Potential Personalized Drug Targets for p53-Deficient Mammary &hellip; <a href=\"https:\/\/www.med.unc.edu\/genetics\/perou-and-collaborators-published-in-disease-models-and-mechanisms\/\" aria-label=\"Read more about Perou and collaborators published in Disease Models and Mechanisms\">Read more<\/a><\/p>\n","protected":false},"author":22429,"featured_media":2773,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"_acf_changed":false,"footnotes":"","_links_to":"","_links_to_target":""},"categories":[2],"tags":[],"class_list":["post-2772","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-news","odd"],"acf":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v26.8 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Perou and collaborators published in Disease Models and Mechanisms | Department of Genetics<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/www.med.unc.edu\/genetics\/perou-and-collaborators-published-in-disease-models-and-mechanisms\/\" \/>\n<meta property=\"og:locale\" content=\"en_US\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Perou and collaborators published in Disease Models and Mechanisms | Department of Genetics\" \/>\n<meta property=\"og:description\" content=\"Charles Perou, PhD, Professor of Genetics and Pathology and Laboratory Medicine and the May Goldman Shaw Distinguished Professor of Molecular Oncology was corresponding author of a study that focused on finding possible drug targets in triple-negative breast cancers. The paper, titled \u201cGenomic Profiling of Murine Mammary Tumors Identifies Potential Personalized Drug Targets for p53-Deficient Mammary &hellip; Read more\" \/>\n<meta property=\"og:url\" content=\"https:\/\/www.med.unc.edu\/genetics\/perou-and-collaborators-published-in-disease-models-and-mechanisms\/\" \/>\n<meta property=\"og:site_name\" content=\"Department of Genetics\" \/>\n<meta property=\"article:published_time\" content=\"2016-09-16T01:34:12+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2018-02-07T16:25:09+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/www.med.unc.edu\/genetics\/wp-content\/uploads\/sites\/481\/2017\/10\/perou-and-collaborators-published-in-disease-models-and-mechanisms-image.jpeg\" \/>\n\t<meta property=\"og:image:width\" content=\"250\" \/>\n\t<meta property=\"og:image:height\" content=\"333\" \/>\n\t<meta property=\"og:image:type\" content=\"image\/jpeg\" \/>\n<meta name=\"author\" content=\"Betsy Clarke\" \/>\n<meta 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